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    SAR156497, an Exquisitely Selective Inhibitor of Aurora Kinases

    Aug 29, 2015

    Jean-Christophe Carry, Franco̧is Clerc, Hervé Minoux, Laurent Schio, Jacques Mauger, Anil Nair, Eric Parmantier, Ronan LeMoigne, Cécile Delorme, Jean-Paul Nicolas, Alain Krick, Pierre-Yves Abećassis, Véronique Crocq-Stuerga, Stéphanie Pouzieux, Laure Delarbre, Sébastien Maignan, Thomas Bertrand, Kirsten Bjergarde, Nina Ma,Sylvette Lachaud, Houlfa Guizani, Reḿi Lebel, Gilles Doerflinger, Sylvie Monget, Sebastien Perron, Francis Gasse, Odile Angouillant-Boniface, Bruno Filoche-Romme,́ Michel Murer, Sylvie Gontier, CeĺinePrev́ost, Marie-Line Monteiro, Cećile Combeau

    A novel selective and orally bioavailable Nav1.8 channel blocker, PF-01247324, attenuates nociception and sensory neuron excitability

    Jan 14, 2015

    Claire Elizabeth Payne, Adam R Brown, Jonathon W Theile, Alexandre J C Loucif, Aristos J Alexandrou, Mathew D Fuller, John H Mahoney, Brett M Antonio, Aaron C Gerlach, David M Printzenhoff, Rebecca L Prime, Gillian Stockbridge, Anthony J Kirkup, Anthony W Bannon, Steve England, Mark L Chapman, Sharan Bagal, Rosemarie Roeloffs, Uma Anand, Praveen Anand, Peter J Bungay, Mark Kemp, Richard P Butt and Edward B Stevens

    Rapid Identification of Metal-Binding Peptoid Oligomers by On-Resin X-Ray Fluorescence Screening

    Jul 18, 2014

    Danielle M. Nalband, Benjamin P. Warner, Nathan H. Zahler, Kent Kirshenbaum

    Voltage sensor interaction site for selective small molecule inhibitors of voltage-gated sodium channels

    Jun 05, 2013

    Ken McCormack, Sonia Santos, Mark L. Chapman, Douglas S. Krafte, Brian E. Marron, Christopher W. West, Michael J. Krambis, Brett M. Antonio, Shannon G. Zellmer, David Printzenhoff, Karen M. Padilla, Zhixin Lin, P. Kay Wagoner, Nigel A. Swain, Paul A. Stupple, Marcel de Groot, Richard P. Butt, and Neil A. Castle

    Discovery of the first non-ATP competitive IGF-1R kinase inhibitors: Advantages in comparison with competitive inhibitors

    Mar 04, 2011

    Dominique Lesuisse, Jacques Mauger, Conception Nemecek, Sébastien Maignan, Janine Boiziau, Greg Harlow, Augustin Hittinger, Swen Ruf, Hartmut Strobel, Anil Nair, Kurt Ritter, Jean-Luc Malleron, Anne Dagallier, Youssef El-Ahmad, Jean-Pierre Guilloteau, Houlfa Guizani, Hervé Bouchard, Corinne Venot

    Voltage-gated potassium channels as therapeutic targets

    Dec 01, 2009

    Heike Wulff, Neil A. Castle and Luis A. Pardo